November 2009
PUBLICATIONS - Back

Biophysics and Biophysical Chemistry Archives

1. Chufán EE, De M, Eipper BA, Mains RE, Amzel LM. Amidation of bioactive peptides:
the structure of the lyase domain of the amidating enzyme. Structure. 2009 Jul15;17(7):965-73.
Key words: enzymes, peptides, lyase
http://www.ncbi.nlm.nih.gov/pubmed/19604476?ordinalpos=3&itool=EntrezSystem2.
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2. Fitzsimmons D, Lukin K, Lutz R, Garvie CW, Wolberger C, Hagman J. Highly cooperative recruitment of Ets-1 and release of autoinhibition by Pax5. J Mol Biol. 2009 Sep 18;392(2):452-64.
Key words: Pax5, proteins, immunology
http://www.ncbi.nlm.nih.gov/pubmed/19616560?ordinalpos=1&itool=EntrezSystem2.
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3. Qiu C, Tarrant MK, Boronina T, Longo PA, Kavran JM, Cole RN, Cole PA, Leahy DJ. In
vitro enzymatic characterization of near full length EGFR in activated and inhibited states. Biochemistry. 2009 Jul 21;48(28):6624-32.
Key words: enzymes, EGFR, biochemistry
http://www.ncbi.nlm.nih.gov/pubmed/19518076?ordinalpos=1&itool=EntrezSystem2.
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1. Chung S, Parker JB, Bianchet M, Amzel LM, Stivers JT. Impact of linker strain and
flexibility in the design of a fragment-based inhibitor. Nat Chem Biol. 2009 Jun;5(6):407-13.
Key words: enzymes, DNA, linkers
http://www.ncbi.nlm.nih.gov/pubmed/19396178?ordinalpos=1&itool=EntrezSystem2.
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2. Hensel Z, Xiao J. A mechanism for stochastic decision making by bacteria. Chembiochem. 2009 Apr 17;10(6):974-6.
Key words: biophysics , fluorescence, gene expression, gene regulation, singlemolecule Studies
http://www.ncbi.nlm.nih.gov/pubmed/19294726?ordinalpos=1&itool=EntrezSystem2.
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1. Acker MG, Shin BS, Nanda JS, Saini AK, Dever TE, Lorsch JR. Kinetic analysis of latesteps of eukaryotic translation initiation. J Mol Biol. 2009 Jan 16;385(2):491-506. Epub 2008 Oct 19.
Key words: eukaryotic translation initiation; protein synthesis; eIF1A
http://www.ncbi.nlm.nih.gov/pubmed/18976658?ordinalpos=3&itool=EntrezSystem2.
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2. Messing SJ, Gabelli SB, Liu Q, Celesnik H, Belasco JG, Piñeiro SA, Amzel LM. Structure and biological function of the RNA Pyrophosphohydrolase BdRppH from Bdellovibrio bacteriovorus. Structure 2009 Mar 11;17(3):472-81.
Key words: RNA, enzymes, bacteria
http://www.ncbi.nlm.nih.gov/pubmed/19278661?ordinalpos=1&itool=EntrezSystem2.
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3. Mustafa AK, van Rossum DB, Patterson RL, Maag D, Ehmsen JT, Gazi SK, Chakraborty A, Barrow RK, Amzel LM, Snyder SH. Glutamatergic regulation of serine racemase via reversal of PIP2 inhibition. Proc Natl Acad Sci U S A. 2009 Feb 24;106(8):2921-6.
Key words: D-serine, metabotropic glutamate receptor, NMDA transmission
http://www.ncbi.nlm.nih.gov/pubmed/19193859?ordinalpos=1&itool=EntrezSystem2.
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4. Shin BS, Kim JR, Acker MG, Maher KN, Lorsch JR, Dever TE. rRNA suppressor of a eukaryotic translation initiation factor 5B/initiation factor 2 mutant reveals a binding site for translational GTPases on the small ribosomal subunit. Mol Cell Biol. 2009 Feb;29(3):808-21. Key words: RNA, ribosomes, proteins
http://www.ncbi.nlm.nih.gov/pubmed/19029250?ordinalpos=10&itool=EntrezSystem2.
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5. Wang T, Yin L, Cooper EM, Lai MY, Dickey S, Pickart CM, Fushman D, Wilkinson KD, Cohen RE, Wolberger C. Evidence for bidentate substrate binding as the basis for the K48 linkage specificity of otubain 1. J Mol Biol. 2009 Mar 6;386(4):1011-23.
Key words: deubiquitination; isopeptide; linkage specificity; otubain
http://www.ncbi.nlm.nih.gov/pubmed/19211026?ordinalpos=1&itool=EntrezSystem2.
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1. Norris A, Bianchet MA, Boeke JD. Compensatory interactions between Sir3p and the nucleosomal LRS surface imply their direct interaction. PLoS Genet. 2008 Dec;4(12):e1000301.
Key words: Sir3p, DNA, telomeres
http://www.ncbi.nlm.nih.gov/pubmed/19079580?ordinalpos=6&itool=EntrezSystem2.
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1. Steyert SR, Messing SAJ, Amzel LM, Gabelli SB, Piñeiro SA. Identification of Bdellovibrio bacteriovorus HD100 Bd0714 as a Nudix dGTPase. J Bacteriol. 2008 Dec;190(24):8215-9
Key words: Bdellovibrio bacteriovorus, bacteria, E. coli
http://www.ncbi.nlm.nih.gov/pubmed/18931106?ordinalpos=1&itool=EntrezSystem2.
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1. Hawse WF, Hoff KG, Fatkins DG, Daines A, Zubkova OV, Schramm VL, Zheng W, Wolberger C. Structural insights into intermediate steps in the Sir2 deacetylation reaction. Structure. 2008 Sep 10;16(9):1368-77.
Key words: deacetylation, Sir2, peptides
http://www.ncbi.nlm.nih.gov/pubmed/18786399?ordinalpos=1&itool=EntrezSystem2.
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2. McLellan JS, Zheng X, Hauk G, Ghirlando R, Beachy PA, Leahy DJ. The mode of Hedgehog binding to Ihog homologues is not conserved across different phyla. Nature, 14 Sep 2008, Letter.
Key words: hedgehog, ihog, proteins
http://www.ncbi.nlm.nih.gov/pubmed/18794898?ordinalpos=1&itool=EntrezSystem2.
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1. Bacha U, Barrila J, Gabelli SB , Kiso Y, Amzel LM and Freire E. Development of broad-spectrum halomethyl ketone inhibitors against coronavirus main protease 3CL(pro). Chem Biol Drug Des. 2008 Jul;72(1):34-49.
Key words: biophysical chemistry, calorimetric techniques, drug design, drug discovery, protease and ligands (substrate/inhibitor)
http://www.ncbi.nlm.nih.gov/pubmed/18611220?ordinalpos=1&itool=EntrezSystem2.
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2. Dong J, Nanda JS, Rahman H, Pruitt MR, Shin B-S, Wong C-M, Lorsch JR ,Hinnebusch AG. Genetic identification of yeast 18S rRNA residues required for efficient recruitment of initiator tRNA(Met) and AUG selection. Genes Dev. 2008 Aug 15;22(16):2242-55.
Key words: GCN4 translational control; rRNA; ribosome; scanning; translation initiation
http://www.ncbi.nlm.nih.gov/pubmed/18708582?ordinalpos=1&itool=EntrezSystem2.
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1. Acker MG, Lorsch JR. Mechanism of ribosomal subunit joining during eukaryotic translation initiation. Biochem Soc Trans. 2008 Aug; 36(Pt 4):653-7.
Key words: ribosomes, eukaryotic
http://www.ncbi.nlm.nih.gov/pubmed/18631135?ordinalpos=1&itool=EntrezSystem2.
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2. Bacha U, Barrila J, Gabelli S, Kisa Y, Amzel LM, Freire E. Development of broad-spectrum halomethyl ketone inhibitors against coronavirus main protease 3CL(pro). Chem Biol Drug Des. 2008 Jul;72(1):34-49.
Key words: ketone, coronavirus, protease 3CL
http://www.ncbi.nlm.nih.gov/pubmed/18611220?ordinalpos=1&itool=EntrezSystem2.
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3. Feeser EA, Wolberger C. Structural and functional studies of the Rap1 C-terminus reveal novel separation-of-function mutants. J Mol Biol. 2008 Jul 11;380(3):520-31.
Key words: Rap 1, C-terminus, mutants
http://www.ncbi.nlm.nih.gov/pubmed/18538788?ordinalpos=1&itool=EntrezSystem2.
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1. Huang CH, Mandelker D, Gabelli SB, Amzel LM. Insights into the oncogenic effects of /PIK3CA/ mutations from the structure of p110alpha/p85alpha. Cell Cycle. 2008 May;7(9):1151-6.
Key words: oncogene, PIK3CA, mutations
http://www.ncbi.nlm.nih.gov/pubmed/18418043?ordinalpos=1&itool=EntrezSystem2.
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2. Mori MX, Vander Kooi CW, Leahy DJ, Yue DT. Crystal structure of the Ca(V)2 IQ domain in complex with Ca(2+)/calmodulin: high-resolution mechanistic implications for channel regulation by Ca(2+). Structure. 2008 Apr;16(4):607-20.
Key words: crystals, structures, calmodulin
http://www.ncbi.nlm.nih.gov/pubmed/18400181?ordinalpos=1&itool=EntrezSystem2.
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1. Bianchet MA, Erdemli SB, Amzel LM. Structure, function, and mechanism of cytosolic quinone reductases.Vitam Horm. 2008;78:63-84.
Key words: Cytosolic, Quinone, Reductases
http://www.ncbi.nlm.nih.gov/pubmed/18374190?ordinalpos=2&itool=EntrezSystem2.
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2. Leahy, D. A molecular view of anti-ErbB monoclonal antibody therapy. Cancer Cell. 2008 Apr;13(4):291-3.
Key words: Anti-ErbB, Antibody
http://www.ncbi.nlm.nih.gov/pubmed/18394550?ordinalpos=2&itool=EntrezSystem2.
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3. Qiu C, Tarrant MK, Choi SH, Sathyamurthy A, Bose R, Banjade S, Pal A, Bornmann WG, Lemmon MA, Cole PA, Leahy DJ. Mechanism of activation and inhibition of the HER4/ErbB4 kinase. Structure. 2008 Mar;16(3):460-7.
Key words: HER4, ErbB4, Kinase
http://www.ncbi.nlm.nih.gov/pubmed/18334220?ordinalpos=2&itool=EntrezSystem2.
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4. Suh Y, Atzmon G, Cho MO, Hwang D, Liu B, Leahy DJ, Barzilai N, Cohen P. Functionally significant insulin-like growth factor I receptor mutations in centenarians. Proc Natl Acad Sci U S A. 2008 Mar 4;105(9):3438-42. Epub 2008 Mar 3.
Key words: Insulin, Centenarians
http://www.ncbi.nlm.nih.gov/pubmed/18316725?ordinalpos=2&itool=EntrezSystem2.
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1. Qiu C, Lienhard S, Hynes NE, Badache A, Leahy DJ. Memo is homologous to nonheme iron dioxygenases and binds an ErbB2-derived phosphopeptide in its vestigial active site. J Biol Chem. 2008 Feb 1;283(5):2734-40. Epub 2007 Nov 28.
Key words: dioxygenases, ErbB2, phosphopeptide, peptides
http://www.ncbi.nlm.nih.gov/pubmed/18045866?ordinalpos=1&itool=EntrezSystem2.
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1. Qiu C, Lienhard S, Hynes NE, Badache A, Leahy DJ. Memo is homologous to nonheme iron dioxygenases and binds an ErbB2-derived phosphopeptide in its vestigial active site. J Biol Chem. 2008 Feb 1;283(5):2734-40. Epub 2007 Nov 28.
Key words: dioxygenases, ErbB2, phosphopeptide, peptides
http://www.ncbi.nlm.nih.gov/pubmed/18045866?ordinalpos=1&itool=EntrezSystem2.
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1. Acker MG, Kolitz SE, Mitchell SF, Nanda JS, Lorsch JR. Reconstitution of yeast translation initiation. Methods Enzymol. 2007;430:111-45.
Key words: Protein Synthesis, mechanism
http://www.ncbi.nlm.nih.gov/pubmed/17913637?ordinalpos=1&itool=EntrezSystem2.
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2. Huang GN, Huso DL, Bouyain S, Tu J, McCorkell KA, May MJ, Zhu Y, Lutz M, Collins S, Dehoff M, Kang S, Whartenby K, Powell J, Leahy D, Worley PF. NFAT binding and regulation of T cell activation by the cytoplasmic scaffolding Homer proteins. Science. 2008 Jan 25;319(5862):476-81.
Key words: NFAT, T cell, Homer
http://www.ncbi.nlm.nih.gov/pubmed/18218901?ordinalpos=1&itool=EntrezSystem2.
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3. Xiao J, Elf J, Li G, Yu J, Xie XS, Imaging gene expression in living cells at the single molecule level. Single Molecules: A Laboratory Manual, edited by Selvin P., and Ta H. Dec. 2007, Cold Spring Harbor Laboratory Press, Cold Spring Harbor, NY.
Key words: Imaging, single molecules

1. Dohán O, Portulano C, Basquin C, Reyna-Neyra A, Amzel LM, Carrasco N. The Na+/I symporter (NIS) mediates electroneutral active transport of the environmental pollutant perchlorate. Proc Natl Acad Sci U S A. 2007 Dec 18;104(51):20250-5.
Key words: plasma membrane protein, perchlorate, pollutants
http://www.ncbi.nlm.nih.gov/pubmed/18077370?ordinalpos=4&itool=EntrezSystem2.
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2. Huang CH, Mandelker D, Schmidt-Kittler O, Samuels Y, Velculescu VE, Kinzler KW, Vogelstein B, Gabelli SB, Amzel LM. The structure of a human p110alpha/p85alpha complex elucidates the effects of oncogenic PI3Kalpha mutations. Science. 2007 Dec14; 318(5857):
1744-8.
Key words: p110alpha/p85alpha; oncogene, mutations, P13Kalpha
http://www.ncbi.nlm.nih.gov/pubmed/18079394?ordinalpos=4&itool=EntrezSystem2.
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3. Leahy DJ. A monkey wrench in the kinase machine. Nat Struct Mol Biol. 2007 Dec;14(12):1120-1.
Key words: kinase,
http://www.ncbi.nlm.nih.gov/pubmed/18059449?ordinalpos=4&itool=EntrezSystem2.
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4. Qiu C, Lienhard S, Hynes NE, Badache A, Leahy DJ. Memo is homologous to nonheme iron dioxygenases and binds an ErbB2-derived phosphopeptide in its vestigial active site. J Biol Chem. 2007 Nov 28; [Epub ahead of print]
Key words: iron dioxygenase, ErbB2, phosphopeptide
http://www.ncbi.nlm.nih.gov/pubmed/18045866?ordinalpos=4&itool=EntrezSystem2.
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November 2009 articles:
Seminar Series
NIH Transformative Research Projects Program
Funding for Prostate Cancer Research
Department of Defense Breast Cancer Research Program (BCRP)
Klarman Family Foundation Grants Program in Eating Disorders Research
Young Investigator Grant for Probiotics Research
The Professor Rahamimoff Travel Grants Program
 
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